SCHEMBL21496790

SCHEMBL21496790

CC1c2ccccc2C(C)(C(N)=O)N1c1nc2ccc(C(F)(F)F)cc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 2/20 0.47
HDAC8 Q9BY41 1/20 0.47
NPY5R Q15761 3/20 0.44
EGLN1 Q9GZT9 1/20 0.43
ALKBH3 Q96Q83 1/20 0.41
LPAR2 Q9HBW0 1/20 0.40
HRH4 Q9H3N8 1/20 0.40
NPBWR1 P48145 1/20 0.39
SLC6A9 P48067 1/20 0.39
ADRA1A P35348 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21496789 0.71 HDAC11 (0.80) HDAC11HDAC8NPY5REGLN1HRH4
SCHEMBL14690446 0.67 HRH4 (0.60) EGLN1HRH4NPBWR1KCNH2SCN10A
SCHEMBL21496730 0.64 HDAC11 (0.81) HDAC11HDAC8NPY5REGLN1ADRA1A
SCHEMBL20132855 0.64 HDAC11 (1.00) HDAC11HDAC8NPY5R
SCHEMBL30468600 0.64 HDAC11 (1.00) HDAC11HDAC8NPY5R
SCHEMBL12280690 0.63 NPY5R (0.52) NPY5RADRA1AKCNH2
SCHEMBL12280688 0.62 NPY5R (0.51) NPY5R
SCHEMBL29153822 0.62 SCN10A (0.49) EGLN1HRH4NPBWR1KCNH2SCN10A
SCHEMBL2421049 0.62 NPY5R (0.63) NPY5RNPBWR1ADRA1AKCNH2
SCHEMBL12281042 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3784654-A1 ISOINDOLINES AS HDAC INHIBITORS Valo Early Discovery, Inc. (US) 2021-03-03 EP disclosed
WO-2019204550-A1 ISOINDOLINES AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2019-10-24 WO disclosed