SCHEMBL2152185

SCHEMBL2152185

CCOc1cccc(-n2cc(C(=O)OC)nc2-c2ccc(F)cc2)c1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 12/20 0.64
GABRA2 P47869 6/20 0.62
GABRB2 P47870 6/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2152511 0.93 GABRA2 (0.73) CCKARGABRA2GABRB2
SCHEMBL2152335 0.89 CCKAR (0.66) CCKARGABRA2GABRB2
SCHEMBL2152521 0.84 GABRA2 (0.75) CCKARGABRA2GABRB2
SCHEMBL2152790 0.82 CCKAR (0.75) CCKAR
SCHEMBL2152420 0.81 CCKAR (0.65) CCKARGABRA2GABRB2
SCHEMBL3133542 0.80 CCKAR (0.63) CCKARGABRA2GABRB2
SCHEMBL2152217 0.80 CCKAR (0.86) CCKAR
SCHEMBL2152132 0.80 CCKAR (0.66) CCKARGABRA2GABRB2
Trifluoroacetic Acid SCHEMBL2203298 0.79 CCKAR (0.70) CCKAR
SCHEMBL3131008 0.78 CCKAR (1.00) CCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010519-B1 SUBSTITUTED IMIDAZOLE 4-CARBOXAMIDES AS CHOLECYSTOKININ-1 RECEPTOR MODULATORS MERCK SHARP & DOHME (US) 2011-07-06 EP disclosed