SCHEMBL21535489

SCHEMBL21535489

Cc1ccsc1[C@@H]1CCN(C)C1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21535638 1.00 KDM4E (0.38) KDM4EATMALDH1A1MEN1GLA
SCHEMBL19995958 0.75 PDE4B (0.43) KDM4EALDH1A1MEN1GAAMAPT
SCHEMBL27522260 0.74 ALDH1A1 (0.37) KDM4EATMALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL4757290 0.71 MAPK1 (0.36) KDM4EALDH1A1GAAMAPTMAPK1
SCHEMBL7431818 0.71 ALDH1A1 (0.39) KDM4EATMALDH1A1MEN1GLA
SCHEMBL5584941 0.69 HTR2C (0.47) KDM4EALDH1A1MEN1GAAMAPT
SCHEMBL19382042 0.69 MAPK1 (0.34) KDM4EALDH1A1MEN1GLAGAA
SCHEMBL15830146 0.68 KDM4E (0.54) KDM4EATM
SCHEMBL10212349 0.68 KDM4E (0.54) KDM4EATM
SCHEMBL17864290 0.68 MAPK1 (0.34) KDM4EALDH1A1MEN1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233858-B1 ERK INHIBITORS MERCK SHARP & DOHME (US) 2019-10-30 EP disclosed