SCHEMBL21546724

SCHEMBL21546724

N#Cc1cccc(-c2cc(-n3c4cc(-c5ncccn5)ccc4c4ccc(-c5ncccn5)cc43)c(C#N)cc2-n2c3cc(-c4ncccn4)ccc3c3ccc(-c4ncccn4)cc32)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 6/20 0.54
CYP1A2 P05177 8/20 0.41
CYP3A4 P08684 7/20 0.41
CYP2D6 P10635 5/20 0.41
CYP2C19 P33261 4/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 3/20 0.41
MAPK1 P28482 2/20 0.41
ALOX15 P16050 1/20 0.41
GRM5 P41594 4/20 0.40
ELANE P08246 2/20 0.39
LMNA P02545 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
TSHR P16473 3/20 0.38
CYP2C9 P11712 2/20 0.38
TP53 P04637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21546725 0.97 CLK4 (0.51) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL21546499 0.92 CLK4 (0.56) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL22760715 0.92 CLK4 (0.46) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL21546611 0.91 CLK4 (0.54) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL21546608 0.91 CLK4 (0.51) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL21546726 0.91 CLK4 (0.51) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL21546631 0.90 ALDH1A3 (0.38) CLK4
SCHEMBL22761048 0.89 CYP1A2 (0.47) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL21546641 0.87 CYP1A2 (0.41) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL22760662 0.86 ALDH1A3 (0.39) CLK4CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3478793-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2019-11-06 EP disclosed