SCHEMBL21548076

SCHEMBL21548076

O=c1[nH]c2ccccc2nc1N1Cc2ccccc2C1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.69
HTR3A P46098 2/20 0.69
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 3/20 0.51
GAA P10253 2/20 0.51
HPGD P15428 2/20 0.51
HSD17B10 Q99714 2/20 0.51
KMT2A Q03164 1/20 0.51
PLAUR Q03405 1/20 0.50
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
PDE10A Q9Y233 1/20 0.47
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
KHK P50053 1/20 0.46
HDAC11 Q96DB2 2/20 0.46
HTT P42858 1/20 0.44
TP53 P04637 1/20 0.44
PYGM P11217 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467563 0.82 HRH4 (1.00) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL31749043 0.81 HRH4 (0.74) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL5237102 0.80 HTR3A (0.72) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL31214382 0.79 HTR3A (0.70) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL31214324 0.79 HRH4 (0.70) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL13801322 0.78 HRH4 (0.72) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL23771247 0.74 HDAC11 (0.63) HTR3ARAB9APDE10ABCHEACHE
SCHEMBL605362 0.74 HRH4 (0.62) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL27563614 0.72 HRH4 (0.62) HRH4HTR3AKDM4EALDH1A1GAA
SCHEMBL5237605 0.69 HRH4 (0.62) HRH4HTR3APDE10ABCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3564240-A1 PIPERIDINE INTERMEDIATES Purdue Pharma L.P. (US) 2019-11-06 EP disclosed