SCHEMBL21550169

SCHEMBL21550169

CCS(=O)(=O)Nc1cc(Br)c(C(=O)c2ccc(F)cc2Cl)cc1F

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
MRGPRX1 Q96LB2 7/20 0.41
HPGD P15428 2/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
PYGL P06737 2/20 0.38
PSIP1 O75475 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
TLR4 O00206 2/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28469745 0.92 KMT2A (0.47) KMT2AMRGPRX1HPGDMAPK13MAPK12
SCHEMBL20157667 0.83 MAPT (0.43) KMT2AMRGPRX1HPGDPSIP1KDM4E
SCHEMBL21564888 0.83 HPGD (0.44) HPGDMAPK13MAPK12MAPK11MAPK14
SCHEMBL20157971 0.81 NPC1 (0.44) KMT2AMRGPRX1HPGDPSIP1KDM4E
SCHEMBL21549994 0.78 HPGD (0.37) KMT2AHPGDMAPK13MAPK12MAPK11
SCHEMBL21550060 0.77 NPC1 (0.38) HPGDMAPK13MAPK12MAPK11MAPK14
SCHEMBL21550021 0.76 MAPK14 (0.45) HPGDMAPK13MAPK12MAPK11MAPK14
SCHEMBL28465102 0.76 MAPK13 (0.44) HPGDMAPK13MAPK12MAPK11MAPK14
SCHEMBL21550148 0.75 PYGL (0.41) HPGDMAPK13MAPK12MAPK11MAPK14
SCHEMBL21550056 0.74 HPGD (0.42) KMT2AHPGDMAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111819181-A Benzo-seven-membered heterocyclic compound, preparation method, pharmaceutical composition and application thereof 罗欣药业(上海)有限公司 2020-10-23 CN disclosed
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed