SCHEMBL2156558

SCHEMBL2156558

O=C(C(=O)c1ccc(O)cc1O)c1ccc(O)cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 1.00
CA12 O43570 5/20 0.70
CA1 P00915 5/20 0.70
CA2 P00918 5/20 0.70
CA7 P43166 5/20 0.70
CA9 Q16790 5/20 0.70
CA14 Q9ULX7 5/20 0.70
ALDH1A1 P00352 2/20 0.70
TSHR P16473 1/20 0.70
HSP90AB1 P08238 1/20 0.59
GFER P55789 1/20 0.59
PDK2 Q15119 1/20 0.59
PDK4 Q16654 1/20 0.59
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
SERPINE1 P05121 1/20 0.57
USP2 O75604 1/20 0.57
GAA P10253 1/20 0.57
KEAP1 Q14145 1/20 0.57
NFE2L2 Q16236 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14641561 0.88 CES2 (0.78) CES2CA12CA1CA2CA7
SCHEMBL14676003 0.86 CES2 (0.75) CES2CA12CA1CA2CA7
SCHEMBL5962551 0.85 CES2 (0.73) CES2CA12CA1CA2CA7
SCHEMBL9263777 0.84 CES2 (0.72) CES2CA12CA1CA2CA7
SCHEMBL29357695 0.84 CES2 (0.73) CES2CA12CA1CA2CA7
SCHEMBL39507 0.84 CES2 (0.73) CES2CA12CA1CA2CA7
SCHEMBL14416852 0.83 CES2 (0.69) CES2CA12CA1CA2CA7
SCHEMBL8906715 0.82 CES2 (0.70) CES2CA12CA1CA2CA7
SCHEMBL5674868 0.82 CES2 (0.70) CES2CA12CA1CA2CA7
2,4-Dihydroxybenzoic Acid SCHEMBL29573604 0.82 CA12 (1.00) CES2CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973034-B2 Ameliorating toxic effects of such as cancer therapy drugs or addictive drug overdose ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2011-07-05 US claimed
US-7996156-B2 Methods for predicting properties of molecules THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-08-09 US disclosed
US-7973034-B2 Ameliorating toxic effects of such as cancer therapy drugs or addictive drug overdose ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2011-07-05 US disclosed
US-7973034-B2 Ameliorating toxic effects of such as cancer therapy drugs or addictive drug overdose ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2011-07-05 US disclosed
US-7973034-B2 Ameliorating toxic effects of such as cancer therapy drugs or addictive drug overdose ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2011-07-05 US disclosed
US-20080146548-A1 AMIDE, ARYL SULFONAMIDE, ARYL UREA, AND a,b-DIKETONE DERIVED CARBOXYLESTERASE INHIBITORS, AND THEIR METHODS OF USE ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2008-06-19 US disclosed
US-20080146548-A1 AMIDE, ARYL SULFONAMIDE, ARYL UREA, AND a,b-DIKETONE DERIVED CARBOXYLESTERASE INHIBITORS, AND THEIR METHODS OF USE ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2008-06-19 US disclosed
US-20080146548-A1 AMIDE, ARYL SULFONAMIDE, ARYL UREA, AND a,b-DIKETONE DERIVED CARBOXYLESTERASE INHIBITORS, AND THEIR METHODS OF USE ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2008-06-19 US disclosed
US-7241551-B2 Positive-working resist composition FUJIFILM CORPORATION (JP) 2007-07-10 US disclosed
US-7241551-B2 Positive-working resist composition FUJIFILM CORPORATION (JP) 2007-07-10 US disclosed
US-20050054691-A1 Carboxylesterase inhibitors ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2005-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054691-A1 Carboxylesterase inhibitors CES1, CES2, BCHE CES2 2/4885CA12 3171/4885CA1 1806/4885
US-20080146548-A1 AMIDE, ARYL SULFONAMIDE, ARYL UREA, AND a,b-DIKETONE DERIVED CARBOXYLESTERASE INHIBITORS, AND THEIR METHODS OF USE CES1, BCHE, CES2 CES2 3/4885CA12 3377/4885CA1 2189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.