SCHEMBL2157454

SCHEMBL2157454

COc1ccc(CCCC(=O)N2CCN(CCOc3ccccc3F)CC2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.50
EBP Q15125 2/20 0.50
TMEM97 Q5BJF2 1/20 0.50
DRD3 P35462 2/20 0.48
DRD2 P14416 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KDM4E B2RXH2 1/20 0.48
EBPL Q9BY08 1/20 0.47
CACNA1F O60840 1/20 0.46
DRD1 P21728 1/20 0.46
DRD4 P21917 1/20 0.46
DRD5 P21918 1/20 0.46
HRH2 P25021 1/20 0.46
ADRA1D P25100 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR7 P34969 1/20 0.46
ADRA1A P35348 1/20 0.46
HRH1 P35367 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2157438 0.93 DRD3 (0.46) SIGMAR1EBPTMEM97DRD3MEN1
SCHEMBL2158498 0.89 SIGMAR1 (0.58) SIGMAR1DRD3DRD2KDM4ECACNA1F
SCHEMBL7032807 0.88 DRD3 (0.53) DRD3DRD2KMT2ACACNA1FDRD1
Hydrochloric Acid SCHEMBL2158183 0.87 DRD3 (0.52) DRD3DRD2CACNA1FDRD1DRD4
SCHEMBL1332065 0.85 SIGMAR1 (0.61) SIGMAR1EBPTMEM97ADRA1DADRA1A
SCHEMBL2158301 0.85 KMT2A (0.57) SIGMAR1DRD3DRD2MEN1KMT2A
SCHEMBL2157909 0.84 KDM4E (0.47) SIGMAR1DRD3MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL2157282 0.84 KMT2A (0.56) DRD3DRD2MEN1KMT2AKDM4E
SCHEMBL2157673 0.83 DRD3 (0.51) SIGMAR1DRD3DRD2CACNA1FDRD1
SCHEMBL2157502 0.81 DRD3 (0.51) SIGMAR1DRD3DRD2KDM4ECACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183374-B2 Piperidine and piperazine derivatives M'S SCIENCE CORPORATION (JP) 2012-05-22 US disclosed
EP-2340835-A1 Piperidine and piperazine derivatives M's Science Corporation (JP) 2011-07-06 EP disclosed
EP-1976525-B1 PIPERIDINE AND PIPERAZINE DERIVATIVES MS SCIENCE CORP (JP) 2010-11-03 EP disclosed