SCHEMBL21583768

SCHEMBL21583768

O=C(CCc1ccc2c(c1)OCCO2)Nc1cccc2cccnc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.65
ALDH1A1 P00352 3/20 0.65
HPGD P15428 2/20 0.65
MEN1 O00255 2/20 0.65
MAPT P10636 2/20 0.65
KMT2A Q03164 2/20 0.65
KDM4E B2RXH2 1/20 0.65
GAA P10253 1/20 0.65
CFTR P13569 1/20 0.57
POLB P06746 1/20 0.56
HTT P42858 1/20 0.54
TDP1 Q9NUW8 1/20 0.52
HDAC6 Q9UBN7 4/20 0.52
HDAC3 O15379 3/20 0.52
HDAC4 P56524 3/20 0.52
HDAC1 Q13547 3/20 0.52
HDAC7 Q8WUI4 3/20 0.52
HDAC2 Q92769 3/20 0.52
HDAC10 Q969S8 3/20 0.52
HDAC11 Q96DB2 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8785242 0.80 POLB (0.60) ALDH1A1HPGDMEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL8781797 0.79 POLB (0.59) ALDH1A1HPGDMEN1MAPTKMT2A
SCHEMBL21565076 0.79 POLB (0.73) RAB9AALDH1A1MEN1MAPTKMT2A
SCHEMBL29894470 0.79 POLB (0.73) RAB9AALDH1A1MEN1MAPTKMT2A
SCHEMBL28561573 0.78 POLB (0.64) RAB9AALDH1A1HPGDMEN1MAPT
SCHEMBL9464627 0.77 POLB (0.88) ALDH1A1HPGDMEN1MAPTKMT2A
SCHEMBL28568043 0.76 MAPT (0.64) RAB9AHPGDMEN1MAPTKMT2A
SCHEMBL29894627 0.76 MAPT (0.64) RAB9AHPGDMEN1MAPTKMT2A
SCHEMBL13676201 0.76 TRPV1 (0.66) ALDH1A1HPGDMEN1MAPTKMT2A
SCHEMBL24803633 0.75 POLB (0.57) RAB9AALDH1A1HPGDMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019228299-A1 SYNTHESIS AND USES OF PEPTIDE BORATE ESTER COMPOUND 江苏正大丰海制药有限公司 (CN) 2019-12-05 WO disclosed