SCHEMBL21584775

SCHEMBL21584775

CN1CCN(C(=O)c2cnco2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA4 P43681 2/20 0.54
CHRNB2 P17787 1/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
CHRNA7 P36544 1/20 0.54
HRH2 P25021 1/20 0.47
HRH1 P35367 1/20 0.47
HRH4 Q9H3N8 5/20 0.46
RIPK1 Q13546 1/20 0.44
POLB P06746 2/20 0.42
CYP1A2 P05177 1/20 0.42
HPGD P15428 2/20 0.42
ATM Q13315 1/20 0.42
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
ALOX15 P16050 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18281138 0.83 CHRNA4 (0.50) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL20152893 0.78 RIPK1 (0.55) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL22874982 0.77 CHRNA4 (0.51) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL18255212 0.76 RIPK1 (0.59) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL20138338 0.75 RIPK1 (0.52) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL21095630 0.74 CHRNA4 (0.62) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL21062061 0.74 CHRNA4 (0.62) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL20935043 0.74 CHRNA4 (0.48) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL15157092 0.73 HRH4 (0.46) HRH4POLBCYP1A2HPGDATM
SCHEMBL18255042 0.72 NPC1 (0.65) POLBHPGDTSHRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019228403-A1 AUTOTAXIN INHIBITORS AND USES THEREOF FRONTHERA U.S. PHARMACEUTICALS LLC (US) 2019-12-05 WO disclosed