SCHEMBL21589368

SCHEMBL21589368

Cn1cc(P(c2ccccc2)c2ccccc2)nn1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 2/20 0.39
GAA P10253 1/20 0.39
BRD4 O60885 2/20 0.36
SLC9A1 P19634 2/20 0.35
KEAP1 Q14145 1/20 0.35
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
NPSR1 Q6W5P4 1/20 0.33
KMT2A Q03164 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
KDM4A O75164 1/20 0.30
KDM5C P41229 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
KDM2A Q9Y2K7 1/20 0.30
KDM3A Q9Y4C1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21589364 0.68 CYP3A4 (0.48) CYP3A4TDP1KDM4EGAABRD4
SCHEMBL28275505 0.67 TDP1 (0.92) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL31412011 0.67 TDP1 (0.92) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL2846416 0.64 TDP1 (0.55) CYP3A4TDP1KDM4EGAAESR1
Ethane SCHEMBL27526681 0.64 TDP1 (0.86) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL2085135 0.64 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL101 0.64 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
Benzene SCHEMBL6890099 0.64 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL5028587 0.64 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
Methyl Alcohol SCHEMBL16974123 0.62 TDP1 (0.80) CYP3A4TDP1KDM4EGAAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019234228-A1 BETA-AMINO-ALPHA-HYDROXYALKYLPHENYL DERIVATIVES AND THEIR USE FOR CANCER TREATMENT RISING TIDE FOUNDATION (CH) 2019-12-12 WO disclosed