SCHEMBL21589433

SCHEMBL21589433

CCSc1nc2ncccc2c(=O)n1CCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3C2A O00443 7/20 0.61
ALDH1A1 P00352 3/20 0.60
POLB P06746 1/20 0.60
CA12 O43570 4/20 0.59
CA2 P00918 4/20 0.59
CA9 Q16790 4/20 0.59
CA1 P00915 3/20 0.59
MAPT P10636 2/20 0.55
PDE4A P27815 1/20 0.54
PDE4B Q07343 1/20 0.54
PDE4C Q08493 1/20 0.54
PDE4D Q08499 1/20 0.54
PIK3C2B O00750 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
LMNA P02545 1/20 0.50
ALDH1A2 O94788 1/20 0.48
ALDH1A3 P47895 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21589401 0.86 PIK3C2A (0.67) PIK3C2AALDH1A1POLBPIK3C2B
SCHEMBL21589376 0.82 PIK3C2A (0.61) PIK3C2AALDH1A1POLBCA12CA2
SCHEMBL21586306 0.76 PIK3C2A (1.00) PIK3C2AMAPTPIK3C2B
SCHEMBL9671550 0.74 PDE7A (0.65) ALDH1A1CA12CA2CA9CA1
SCHEMBL21589406 0.74 PIK3C2A (0.65) PIK3C2AALDH1A1MAPTPIK3C2BALDH1A2
SCHEMBL5921047 0.73 CASR (0.74) MEN1KMT2A
SCHEMBL21589398 0.72 PIK3C2A (0.65) PIK3C2APIK3C2B
SCHEMBL6512906 0.72 PDE4A (0.86) ALDH1A1MAPTPDE4APDE4BPDE4C
SCHEMBL30003002 0.70 PIK3C2A (0.74) PIK3C2APIK3C2B
SCHEMBL21586276 0.70 PIK3C2A (0.81) PIK3C2AALDH1A1POLBMAPTPIK3C2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019234237-A1 HETEROCYCLIC COMPOUNDS AS CLASS II PHOSPHOINOSITIDE 3-KINASE INHIBITORS FORSCHUNGSVERBUND BERLIN E.V. (DE) 2019-12-12 WO disclosed