SCHEMBL21589693

SCHEMBL21589693

CCCCC1(CC)CN(c2ccccc2)c2cc(Br)c(O)cc2SN1C

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.31
KDM4E B2RXH2 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21589670 0.86 DRD2 (0.31) ELANE
SCHEMBL21589621 0.86 NR1H4 (0.33) ELANE
SCHEMBL24940647 0.80
SCHEMBL30912778 0.78 ELANE (0.32) ELANEKDM4EPKM
SCHEMBL21585962 0.78 ELANE (0.32) ELANEKDM4EPKM
SCHEMBL8333225 0.78 ELANE (0.31) ELANEKDM4EPKM
SCHEMBL8330763 0.78 ELANE (0.31) ELANEKDM4EPKM
SCHEMBL21589493 0.78 NR1H4 (0.32) ELANEKDM4EPKM
SCHEMBL24940626 0.73 NR1H4 (0.35)
SCHEMBL19848461 0.72 ELANE (0.33) ELANEKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802504-B1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2023-01-18 EP disclosed
WO-2019234077-A1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2019-12-12 WO disclosed