SCHEMBL21590213

SCHEMBL21590213

Cc1cc([N+](=O)[O-])ccc1N(C)CCN(C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.55
TDP1 Q9NUW8 2/20 0.51
TSHR P16473 2/20 0.51
CYP3A4 P08684 4/20 0.49
HTT P42858 2/20 0.44
TP53 P04637 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNA4 P43681 1/20 0.44
PDE2A O00408 1/20 0.44
PDE5A O76074 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
APEX1 P27695 1/20 0.44
PDE4A P27815 1/20 0.44
BLM P54132 1/20 0.44
PDE1B Q01064 1/20 0.44
PMP22 Q01453 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE7A Q13946 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30221438 0.84 ALDH1A1 (0.51) ALDH1A1TDP1TSHRHTTTP53
SCHEMBL24900387 0.84 ALDH1A1 (0.51) ALDH1A1TDP1TSHRHTTTP53
SCHEMBL3054692 0.84 ALDH1A1 (0.51) ALDH1A1TDP1TSHRCYP3A4HTT
SCHEMBL28462224 0.83 ALDH1A1 (0.53) ALDH1A1TSHRHTTTP53CHRNB2
SCHEMBL3057834 0.83 ALDH1A1 (0.50) ALDH1A1CYP3A4HTTTP53CHRNB2
SCHEMBL24900389 0.83 ALDH1A1 (0.50) ALDH1A1TDP1TSHRHTTTP53
SCHEMBL18030205 0.83 ALDH1A1 (0.50) ALDH1A1TDP1TSHRCYP3A4HTT
SCHEMBL4749290 0.82 ERN1 (0.50) ALDH1A1TDP1HTTTP53CHRNB2
SCHEMBL24900594 0.81 ALDH1A1 (0.48) ALDH1A1TDP1TSHRHTTTP53
SCHEMBL4749269 0.81 ALDH1A1 (0.54) ALDH1A1HTTTP53CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed