SCHEMBL21592544

SCHEMBL21592544

CN(C)CCN1CCN(C(=O)c2ccc(-c3c[nH]c4ncc(-c5ccc(N6CCN(C)CC6)cc5)nc34)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 6/20 0.67
MAP3K11 Q16584 3/20 0.44
CHEK1 O14757 4/20 0.42
PRKD1 Q15139 1/20 0.42
JAK2 O60674 1/20 0.41
ATR Q13535 1/20 0.41
CLK1 P49759 1/20 0.41
DYRK1A Q13627 1/20 0.41
MAPK1 P28482 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
CCNE2 O96020 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21592620 0.87 MAP4K1 (0.64) MAP4K1MAP3K11CHEK1ATR
SCHEMBL21592436 0.86 MAP4K1 (0.64) MAP4K1MAP3K11CHEK1JAK2CLK1
SCHEMBL21592624 0.85 MAP4K1 (0.83) MAP4K1CHEK1PRKD1ATRCLK1
SCHEMBL21592467 0.85 MAP3K11 (0.60) MAP4K1MAP3K11CLK1DYRK1A
SCHEMBL21592553 0.85 MAP4K1 (0.65) MAP4K1MAP3K11CHEK1JAK2ATR
SCHEMBL21592653 0.85 MAP4K1 (0.72) MAP4K1CHEK1PRKD1JAK2CLK1
SCHEMBL21592494 0.84 MAP4K1 (0.81) MAP4K1CHEK1PRKD1ATRCLK1
SCHEMBL21592435 0.83 MAP4K1 (0.77) MAP4K1CHEK1CLK1DYRK1AMAPK1
SCHEMBL28509578 0.82 MAP4K1 (0.70) MAP4K1CHEK1CLK1DYRK1AMAPK1
SCHEMBL21592754 0.82 MAP4K1 (0.68) MAP4K1CHEK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed