SCHEMBL21593058

SCHEMBL21593058

Cc1cc(-c2c[nH]c3ncc(-c4cc(C)c(N5CCN(C)CC5)c(C)c4)nc23)ccc1C(=O)N(C)C

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 8/20 0.74
TNIK Q9UKE5 1/20 0.41
MAPK1 P28482 5/20 0.41
JAK2 O60674 3/20 0.40
JAK1 P23458 3/20 0.40
TYK2 P29597 3/20 0.40
JAK3 P52333 3/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
CAMKK2 Q96RR4 1/20 0.38
MAP3K11 Q16584 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22922391 0.94 MAP4K1 (0.68) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL21592719 0.92 MAP4K1 (0.63) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL22922490 0.86 MAP4K1 (0.58) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL21592752 0.86 MAP4K1 (0.55) MAP4K1MAPK1JAK2JAK1TYK2
SCHEMBL21592732 0.86 MAP4K1 (0.64) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL21592772 0.85 MAP4K1 (0.55) MAP4K1MAPK1JAK2JAK1TYK2
SCHEMBL22858757 0.85 MAP4K1 (1.00) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL29607707 0.85 MAP4K1 (1.00) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL22858850 0.85 MAP4K1 (0.88) MAP4K1TNIKMAPK1JAK2JAK1
SCHEMBL29609216 0.85 MAP4K1 (0.88) MAP4K1TNIKMAPK1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed