SCHEMBL21593676

SCHEMBL21593676

CNc1cnc(Cl)nc1NC1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
AXL P30530 2/20 0.41
FLT3 P36888 1/20 0.40
CYP1A2 P05177 5/20 0.40
MEN1 O00255 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP3A4 P08684 1/20 0.40
BRD4 O60885 2/20 0.39
ATAD2 Q6PL18 2/20 0.39
IKBKB O14920 1/20 0.39
CLK4 Q9HAZ1 2/20 0.38
TYRO3 Q06418 2/20 0.38
SELP P16109 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
HSD17B10 Q99714 2/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
HIF1A Q16665 1/20 0.37
CTSC P53634 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177285 0.87 KMT2A (0.61) KMT2AAXLMEN1HSD17B10
SCHEMBL20329963 0.83 MAPK1 (0.48) KMT2AAXLTYRO3SELP
SCHEMBL21593636 0.83 KMT2A (0.47) KMT2AAXLFLT3TYRO3MERTK
SCHEMBL17196933 0.82 KMT2A (0.51) KMT2AAXLFLT3CYP1A2MEN1
SCHEMBL21593667 0.82 KMT2A (0.46) KMT2AAXL
SCHEMBL20330322 0.81 KMT2A (0.45) KMT2AAXL
SCHEMBL1783841 0.79 KMT2A (0.49) KMT2AAXLFLT3CYP1A2MEN1
SCHEMBL12526937 0.79 KMT2A (0.73) KMT2AAXLCYP1A2MEN1CYP2D6
SCHEMBL12526913 0.79 NSD2 (0.46) KMT2AAXLCYP1A2MEN1CYP2D6
Hydrochloric Acid SCHEMBL1748456 0.78 KMT2A (0.71) KMT2AAXLCYP1A2MEN1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805400-A Dihydropurine thioketone derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-07-29 CN disclosed
WO-2019238929-A1 PURINONE COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2019-12-19 WO disclosed