SCHEMBL21596321

SCHEMBL21596321

CC(O)CNc1cc(Cl)ncc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.41
JAK3 P52333 4/20 0.39
JAK2 O60674 4/20 0.39
JAK1 P23458 3/20 0.39
TYK2 P29597 3/20 0.39
IRAK4 Q9NWZ3 2/20 0.39
SIRT6 Q8N6T7 1/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KCNH2 Q12809 5/20 0.36
ATM Q13315 5/20 0.36
ATR Q13535 3/20 0.36
SYK P43405 2/20 0.36
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDR P35968 1/20 0.36
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30379577 1.00 NNMT (0.41) NNMTJAK3JAK2JAK1TYK2
SCHEMBL18341498 0.87 MEN1 (0.43) IRAK4MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL21600910 0.83 NNMT (0.37) NNMTJAK3JAK2JAK1TYK2
SCHEMBL29127194 0.82 MKNK1 (0.48) NNMTJAK3JAK2JAK1TYK2
SCHEMBL30664056 0.82 MKNK1 (0.48) NNMTJAK3JAK2JAK1TYK2
SCHEMBL21389883 0.82 GAA (0.53) IRAK4MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL16873076 0.82 GAA (0.53) IRAK4MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL15110184 0.80 IRAK4 (0.46) NNMTJAK3JAK2JAK1TYK2
SCHEMBL12411786 0.78 NNMT (0.41) NNMTJAK3JAK2JAK1TYK2
SCHEMBL30678683 0.77 NNMT (0.57) NNMTJAK3JAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112313207-B Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2023-02-14 CN disclosed
CN-112313207-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-02-02 CN disclosed
WO-2019242689-A1 CYANO-SUBSTITUTED PYRIDINE AND CYANO-SUBSTITUTED PYRIMIDINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2019-12-26 WO disclosed
WO-2019242689-A1 CYANO-SUBSTITUTED PYRIDINE AND CYANO-SUBSTITUTED PYRIMIDINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2019-12-26 WO disclosed