SCHEMBL21621426

SCHEMBL21621426

COc1nn(C2CCCCO2)cc1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.36
CD274 Q9NZQ7 1/20 0.35
ABL1 P00519 1/20 0.35
SLC6A3 Q01959 2/20 0.34
ATR Q13535 4/20 0.34
POLQ O75417 1/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
AR P10275 1/20 0.32
CYP4F2 P78329 2/20 0.32
CYP4A11 Q02928 2/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
FLT3 P36888 1/20 0.31
SYK P43405 1/20 0.31
AURKB Q96GD4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21621425 0.84 LMNA (0.38) MAPK1CD274ABL1TDP1
SCHEMBL5122723 0.83 ABL1 (0.38) CD274ABL1ATRCYP4F2CYP4A11
SCHEMBL28479530 0.81 ATR (0.36) CD274ABL1ATRPOLBCYP4F2
SCHEMBL16057646 0.80 ABL1 (0.36) CD274ABL1ATRPOLBCYP4F2
SCHEMBL15634393 0.79 ATR (0.35) CD274ABL1ATRRXRARXRB
SCHEMBL32684090 0.79 CYP2C19 (0.33) CD274ABL1CYP4F2CYP4A11FLT3
SCHEMBL21570191 0.78 POLB (0.39) POLBTDP1BTK
SCHEMBL22235605 0.77 ELANE (0.39) ABL1POLB
SCHEMBL18209667 0.77 ATR (0.36) CD274ABL1ATRCYP4F2CYP4A11
SCHEMBL25189905 0.76 CD274 (0.36) CD274ABL1CYP4F2CYP4A11RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020011254-A1 FUSED TRI-CYCLIC COMPOUND AS PDE3/PDE4 DUAL INHIBITOR 正大天晴药业集团股份有限公司 2020-01-16 WO disclosed