SCHEMBL21622830

SCHEMBL21622830

c1cnc2c(c1)ccc1cccc(-c3ccc4oc5ccc(-c6cccc7ccc8cccnc8c67)cc5c4c3)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.44
CCR8 P51685 5/20 0.44
CCR5 P51681 3/20 0.44
MAPT P10636 3/20 0.44
LMNA P02545 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MMP2 P08253 2/20 0.44
TSHR P16473 2/20 0.44
GMNN O75496 1/20 0.44
TP53 P04637 1/20 0.44
HSP90AA1 P07900 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MMP9 P14780 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
MMP8 P22894 1/20 0.44
THPO P40225 1/20 0.44
MTOR P42345 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21622822 0.94 PIM1 (0.41) CCR1CCR8CCR5MAPTLMNA
SCHEMBL21622503 0.93 CCR1 (0.38) CCR1CCR8CCR5MAPTLMNA
SCHEMBL16629661 0.93 HTT (0.38) CCR1CCR8CCR5MAPTLMNA
SCHEMBL21622500 0.92 KDM4E (0.37) CCR1CCR8CCR5MAPTLMNA
SCHEMBL21622577 0.91 ALOX5 (0.40) CCR1CCR8CCR5MAPTLMNA
SCHEMBL21622684 0.91 HCRTR1 (0.40) CCR1CCR8CCR5MAPTLMNA
SCHEMBL21622506 0.90 MAPT (0.40) CCR1CCR8CCR5MAPTLMNA
SCHEMBL24926017 0.89 BRD4 (0.38) CCR1CCR8CCR5MAPTLMNA
SCHEMBL24926020 0.89 MAPT (0.38) CCR1CCR8CCR5MAPTLMNA
SCHEMBL24927081 0.89 GRM4 (0.36) CCR1CCR8CCR5MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3820965-B1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2023-01-25 EP disclosed
WO-2020011658-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2020-01-16 WO disclosed