SCHEMBL21634804

SCHEMBL21634804

O=C1O[C@@H](Cn2ccnn2)CN1c1cc(F)c(N2CCC(C3CS(O)(O)C3)CC2)c(F)c1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 17/20 0.56
MAOB P27338 1/20 0.56
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 1/20 0.53
KCNH2 Q12809 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21634806 1.00 MAOA (0.56) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL21634805 0.92 MAOA (0.56) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL28562144 0.92 MAOA (0.56) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL21634836 0.90 MAOA (0.61) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL21634838 0.90 MAOA (0.61) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL21634794 0.89 MAOA (0.72) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL4171317 0.84 MAOA (0.60) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL21635096 0.84 MAOA (0.56) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL4883403 0.83 MAOA (0.58) MAOAMAOBCYP3A4CYP2D6KCNH2
SCHEMBL18410309 0.83 MAOA (0.77) MAOAMAOBCYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020021468-A1 SUBSTITUTED OXAZOLIDINONES FOR THE TREATMENT OF MAMMALIAN INFECTIONS CADILA HEALTHCARE LIMITED (IN) 2020-01-30 WO claimed
WO-2020021468-A1 SUBSTITUTED OXAZOLIDINONES FOR THE TREATMENT OF MAMMALIAN INFECTIONS CADILA HEALTHCARE LIMITED (IN) 2020-01-30 WO disclosed