SCHEMBL2164292

SCHEMBL2164292

CCCCOc1cc2nnnc(Nc3ccc(Cl)c(Cl)c3)c2cc1OC

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.60
KDR P35968 17/20 0.58
EPHA2 P29317 16/20 0.58
EPHB4 P54760 13/20 0.58
ERBB2 P04626 5/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2164464 0.97 EGFR (0.64) EGFRKDREPHA2EPHB4ERBB2
SCHEMBL2163104 0.93 EPHA2 (0.56) EGFRKDREPHA2EPHB4ERBB2
SCHEMBL2164519 0.91 EGFR (0.73) EGFRKDREPHB4ERBB2
SCHEMBL2163808 0.90 EPHA2 (0.57) EGFRKDREPHA2EPHB4ERBB2
SCHEMBL2164438 0.89 KDR (0.61) EGFRKDR
SCHEMBL2163102 0.88 EGFR (0.78) EGFRKDREPHB4ERBB2
SCHEMBL2163884 0.87 EGFR (0.63) EGFRKDREPHA2ERBB2
SCHEMBL2165623 0.86 EGFR (0.61) EGFRKDR
SCHEMBL2164453 0.86 KDR (0.53) EGFRKDR
SCHEMBL2162990 0.86 SRC (0.55) EGFRKDREPHA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8349835-B2 Aromatic ring fused triazine derivatives and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2013-01-08 US claimed
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2011-07-28 US claimed
EP-2251332-A1 THE AROMATIC RING TRIAZINE DERIVATIVES AND THE USES THEREOF Shenyang Pharmaceutical University (CN) 2010-11-17 EP claimed
US-8349835-B2 Aromatic ring fused triazine derivatives and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2013-01-08 US disclosed
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2011-07-28 US disclosed
EP-2251332-A1 THE AROMATIC RING TRIAZINE DERIVATIVES AND THE USES THEREOF Shenyang Pharmaceutical University (CN) 2010-11-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF KDR, FLT1, FLT4 EGFR 8/4885KDR 1/4885EPHA2 625/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.