SCHEMBL2164464

SCHEMBL2164464

CCCCCOc1cc2nnnc(Nc3ccc(Cl)c(Cl)c3)c2cc1OC

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.64
EPHA2 P29317 17/20 0.57
KDR P35968 17/20 0.57
EPHB4 P54760 14/20 0.57
ERBB2 P04626 4/20 0.56
FLT1 P17948 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2164292 0.97 EGFR (0.60) EGFREPHA2KDREPHB4ERBB2
SCHEMBL2163104 0.92 EPHA2 (0.56) EGFREPHA2KDREPHB4ERBB2
SCHEMBL2163102 0.91 EGFR (0.78) EGFRKDREPHB4ERBB2
SCHEMBL2165623 0.90 EGFR (0.61) EGFRKDRFLT1
SCHEMBL2163808 0.89 EPHA2 (0.57) EGFREPHA2KDREPHB4ERBB2
SCHEMBL2164519 0.88 EGFR (0.73) EGFRKDREPHB4ERBB2
SCHEMBL2164536 0.87 EGFR (0.62) EGFREPHA2KDRERBB2FLT1
SCHEMBL2164438 0.86 KDR (0.61) EGFRKDRFLT1
SCHEMBL2165852 0.86 EGFR (0.54) EGFRKDR
SCHEMBL2163530 0.86 EGFR (0.56) EGFREPHA2KDRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8349835-B2 Aromatic ring fused triazine derivatives and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2013-01-08 US claimed
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2011-07-28 US claimed
EP-2251332-A1 THE AROMATIC RING TRIAZINE DERIVATIVES AND THE USES THEREOF Shenyang Pharmaceutical University (CN) 2010-11-17 EP claimed
US-8349835-B2 Aromatic ring fused triazine derivatives and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2013-01-08 US disclosed
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2011-07-28 US disclosed
EP-2251332-A1 THE AROMATIC RING TRIAZINE DERIVATIVES AND THE USES THEREOF Shenyang Pharmaceutical University (CN) 2010-11-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF KDR, FLT1, FLT4 EGFR 8/4885EPHA2 625/4885KDR 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.