SCHEMBL2164413

SCHEMBL2164413

CCOc1cc2nnnc(Nc3cc(F)cc(F)c3)c2cc1OC

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.53
KDR P35968 2/20 0.52
RET P07949 1/20 0.52
KIF5B P33176 1/20 0.52
SRC P12931 3/20 0.51
FBP1 P09467 2/20 0.51
EPHA2 P29317 1/20 0.47
EPHB4 P54760 1/20 0.47
LCK P06239 2/20 0.46
CSF1R P07333 1/20 0.44
GAK O14976 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2164707 0.90 SRC (0.55) EGFRKDRRETKIF5BSRC
SCHEMBL2163510 0.89 SRC (0.54) EGFRKDRRETKIF5BSRC
SCHEMBL2164281 0.87 KDR (0.49) EGFRKDRRETKIF5BSRC
SCHEMBL2164488 0.86 SRC (0.51) EGFRKDRSRCFBP1EPHA2
SCHEMBL2165397 0.84 EGFR (0.60) EGFRKDRRETSRCFBP1
SCHEMBL2164111 0.83 SLC2A1 (0.55) EGFRKDRRETSRCLCK
SCHEMBL2164278 0.83 KDR (0.45) EGFRKDRRETKIF5BSRC
SCHEMBL2164641 0.82 FBP1 (0.69) EGFRKDRFBP1EPHB4
SCHEMBL2164632 0.82 EGFR (0.51) EGFRKDRRETKIF5BFBP1
SCHEMBL2163779 0.82 KDR (0.61) EGFRKDRSRCFBP1EPHB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8349835-B2 Aromatic ring fused triazine derivatives and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2013-01-08 US claimed
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2011-07-28 US claimed
EP-2251332-A1 THE AROMATIC RING TRIAZINE DERIVATIVES AND THE USES THEREOF Shenyang Pharmaceutical University (CN) 2010-11-17 EP claimed
US-8349835-B2 Aromatic ring fused triazine derivatives and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2013-01-08 US disclosed
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2011-07-28 US disclosed
EP-2251332-A1 THE AROMATIC RING TRIAZINE DERIVATIVES AND THE USES THEREOF Shenyang Pharmaceutical University (CN) 2010-11-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183972-A1 AROMATIC RING FUSED TRIAZINE DERIVATIVES AND USES THEREOF KDR, FLT1, FLT4 EGFR 8/4885KDR 1/4885RET 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.