SCHEMBL2164733

SCHEMBL2164733

Nc1nc(N)c2c(OCC3CCN(C(=O)c4ccco4)CC3)cccc2n1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DCPS Q96C86 15/20 0.69
DHFR P00374 2/20 0.59
CYP2D6 P10635 1/20 0.54
HIF1A Q16665 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
RCE1 Q9Y256 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2166003 0.85 DCPS (0.81) DCPSDHFRCYP2D6
SCHEMBL2164637 0.84 DCPS (0.75) DCPSDHFRCYP2D6
SCHEMBL2166718 0.83 DCPS (0.71) DCPSDHFRCYP2D6
SCHEMBL2164721 0.83 DCPS (0.74) DCPSDHFRCYP2D6
SCHEMBL1155318 0.83 DCPS (0.74) DCPSDHFRCYP2D6
SCHEMBL2165373 0.83 DCPS (0.72) DCPSDHFRCYP2D6
SCHEMBL1154905 0.83 DCPS (0.74) DCPSDHFRCYP2D6
SCHEMBL2166197 0.83 DCPS (0.71) DCPSDHFRCYP2D6
SCHEMBL2165530 0.83 DCPS (0.71) DCPSDHFRCYP2D6
SCHEMBL2164648 0.82 DCPS (0.70) DCPSDHFRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7985755-B2 2,4-diaminoquinazolines for spinal muscular atrophy FAMILIES OF SPINAL MUSCULAR ATROPHY (US) 2011-07-26 US claimed