SCHEMBL21650784

SCHEMBL21650784

COc1cc(N)ccc1C(=O)N1CCN(C)CC1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
HPGD P15428 2/20 0.61
POLB P06746 1/20 0.52
HTT P42858 2/20 0.51
LMNA P02545 2/20 0.51
TSHR P16473 2/20 0.51
HRH4 Q9H3N8 5/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
GFER P55789 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7154189 0.88 MEN1 (0.65) ALDH1A1HPGDHTTLMNATSHR
SCHEMBL10156660 0.87 HPGD (0.67) ALDH1A1HPGDPOLBHTTLMNA
SCHEMBL7503096 0.86 ALDH1A1 (0.56) ALDH1A1HPGDHTTLMNATSHR
SCHEMBL18753369 0.85 ALDH1A1 (0.52) ALDH1A1HPGDHTTLMNATSHR
SCHEMBL22172135 0.85 ALDH1A1 (0.52) ALDH1A1HPGDPOLBHTTLMNA
SCHEMBL15651032 0.84 ALDH1A1 (0.60) ALDH1A1HPGDPOLBLMNATSHR
SCHEMBL18754001 0.84 ALDH1A1 (0.55) ALDH1A1HPGDHTTLMNATSHR
SCHEMBL7871104 0.84 HPGD (0.63) ALDH1A1HPGDPOLBHTTLMNA
SCHEMBL1447972 0.84 ALDH1A1 (0.63) ALDH1A1HPGDPOLBHTTLMNA
SCHEMBL3925726 0.84 HTT (0.55) ALDH1A1HPGDPOLBHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3241554-B1 QUINOLINE-8-SULFONAMIDE DERIVATIVES HAVING AN ANTICANCER ACTIVITY AGIOS PHARMACEUTICALS INC (US) 2020-01-29 EP disclosed