SCHEMBL2165484

SCHEMBL2165484

CC(C)(C)c1ccc(S(=O)(=O)N2CCC(COc3cccc4nc(N)nc(N)c34)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DCPS Q96C86 15/20 0.60
DHFR P00374 2/20 0.56
CYP2D6 P10635 1/20 0.54
MCHR1 Q99705 1/20 0.48
HSD11B1 P28845 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2166434 0.91 DCPS (0.65) DCPSDHFRCYP2D6
SCHEMBL2166475 0.90 DCPS (0.63) DCPSDHFRCYP2D6
SCHEMBL2167314 0.90 DCPS (0.63) DCPSDHFRCYP2D6
SCHEMBL2164565 0.89 DCPS (0.64) DCPSDHFRCYP2D6
SCHEMBL2164750 0.89 DCPS (0.70) DCPSDHFRCYP2D6
SCHEMBL2164724 0.88 DCPS (0.69) DCPSDHFRCYP2D6
SCHEMBL2168994 0.87 DCPS (0.63) DCPSDHFRCYP2D6
SCHEMBL2166694 0.86 DCPS (0.63) DCPSDHFRCYP2D6
SCHEMBL2166305 0.85 DCPS (0.66) DCPSDHFRCYP2D6
SCHEMBL2166806 0.84 DCPS (0.64) DCPSDHFRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7985755-B2 2,4-diaminoquinazolines for spinal muscular atrophy FAMILIES OF SPINAL MUSCULAR ATROPHY (US) 2011-07-26 US claimed