SCHEMBL21660459

SCHEMBL21660459

N#Cc1ccc2nc(Cl)c(C(=O)O)c(N)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.45
POLB P06746 1/20 0.36
RECQL P46063 1/20 0.36
CASP6 P55212 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CASP1 P29466 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MTOR P42345 1/20 0.36
PIK3CG P48736 1/20 0.36
PRKDC P78527 1/20 0.36
ATM Q13315 1/20 0.36
ATR Q13535 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC22A12 Q96S37 2/20 0.36
HTR1A P08908 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23319181 0.81 NCEH1 (0.35) PIN1POLBPIK3CAPIK3CBMTOR
SCHEMBL15131951 0.75 NCEH1 (0.42) PIN1ALDH1A1DYRK1AKMT2A
SCHEMBL5565734 0.72 PIN1 (0.48) PIN1SLC22A12DYRK1AKMT2AAPP
SCHEMBL9330478 0.72 PIN1 (0.48) PIN1ATMALDH1A1MAPK1SMN1; SMN2
SCHEMBL19876633 0.70 HTT (0.58) PIN1CA1CA2APPMAP4K4
SCHEMBL7505331 0.69 PIN1 (0.40) PIN1ALDH1A1CA1CA2APP
SCHEMBL31401848 0.69 PIN1 (0.41) PIN1L3MBTL1ALDH1A1SLC22A12KMT2A
SCHEMBL11458292 0.69 CA1 (0.50) PIN1ATMALDH1A1KMT2ACA1
SCHEMBL22833509 0.69 ADORA2A (0.50) PIN1PRKDCATRALDH1A1MAPK1
SCHEMBL121243 0.68 APP (0.40) PIN1ALDH1A1PKMYT1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3022205-B1 NOVEL PHOSPHODIESTERASE INHIBITORS AND USES THEREOF UNIV COLUMBIA (US) 2020-02-05 EP disclosed