SCHEMBL21661365

SCHEMBL21661365

CC1CN(c2ccc(C(F)(F)F)c3ncccc23)CC(CN2CCC(N3CCOCC3)CC2)O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
RAD52 P43351 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NCF1 P14598 1/20 0.37
TLR7 Q9NYK1 6/20 0.36
TLR9 Q9NR96 5/20 0.36
TLR8 Q9NR97 5/20 0.36
HTR1A P08908 6/20 0.33
TRPV1 Q8NER1 2/20 0.33
SLC40A1 Q9NP59 1/20 0.33
CLK2 P49760 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CSNK2A1 P68400 1/20 0.33
STK3 Q13188 1/20 0.33
HIPK4 Q8NE63 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
USP2 O75604 1/20 0.33
TP53 P04637 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21661354 1.00 KDM4E (0.37) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL21661470 0.93 KDM4E (0.38) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL16633863 0.86 TLR9 (0.48) KDM4ERAD52L3MBTL1TLR7TLR9
SCHEMBL16633866 0.86 TLR9 (0.48) KDM4ERAD52L3MBTL1TLR7TLR9
SCHEMBL21661609 0.85 NCF1 (0.41) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL21661610 0.85 NCF1 (0.41) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL18980379 0.85 TLR7 (0.40) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL18980767 0.85 TLR7 (0.40) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL29722322 0.85 TLR7 (0.40) KDM4ERAD52L3MBTL1NCF1TLR7
SCHEMBL18980381 0.85 TLR7 (0.40) KDM4ERAD52L3MBTL1NCF1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020025517-A1 TLR7/8 ANTAGONISTS AND USES THEREOF MERCK PATENT GMBH (DE) 2020-02-06 WO disclosed