SCHEMBL21661577

SCHEMBL21661577

Cc1c(F)cc(N2CC(C)O[C@@H](CN3CCC(N4CCCC4)CC3)C2)c2cccnc12

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
RAD52 P43351 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTR1A P08908 10/20 0.37
HRH3 Q9Y5N1 3/20 0.35
TLR9 Q9NR96 3/20 0.34
TLR8 Q9NR97 3/20 0.34
TLR7 Q9NYK1 3/20 0.34
HTT P42858 1/20 0.34
ALK Q9UM73 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21661576 1.00 KDM4E (0.37) KDM4ERAD52L3MBTL1HTR1AHRH3
SCHEMBL21661470 0.84 KDM4E (0.38) KDM4ERAD52L3MBTL1HTR1AHRH3
SCHEMBL16633859 0.81 TLR9 (0.49) KDM4ERAD52L3MBTL1HRH3TLR9
SCHEMBL16633862 0.81 TLR9 (0.49) KDM4ERAD52L3MBTL1HRH3TLR9
SCHEMBL23893140 0.81 HRH3 (0.39) KDM4ERAD52L3MBTL1HTR1AHRH3
SCHEMBL21645266 0.81 KDM4E (0.40) KDM4EL3MBTL1HTT
SCHEMBL21661509 0.81 KDM4E (0.40) KDM4EL3MBTL1HTT
SCHEMBL21661052 0.81 KDM4E (0.40) KDM4EL3MBTL1HTT
SCHEMBL16634343 0.81 TLR8 (0.48) KDM4ERAD52L3MBTL1HRH3TLR9
SCHEMBL24404851 0.81 TLR8 (0.48) KDM4ERAD52L3MBTL1HRH3TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020025517-A1 TLR7/8 ANTAGONISTS AND USES THEREOF MERCK PATENT GMBH (DE) 2020-02-06 WO disclosed