SCHEMBL23893140

SCHEMBL23893140

Cc1ccc(N2C[C@H](CN3CCC(N4CCCC4)CC3)O[C@H](C)C2)c2nccnc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.39
KDM4E B2RXH2 2/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
TLR9 Q9NR96 3/20 0.33
TLR8 Q9NR97 3/20 0.33
TLR7 Q9NYK1 3/20 0.33
HTR1A P08908 4/20 0.33
RAD52 P43351 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MBTD1 Q05BQ5 1/20 0.31
L3MBTL3 Q96JM7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18980659 0.88 HRH3 (0.39) HRH3KDM4EHTTKMT2ARAD52
SCHEMBL21661451 0.88 TLR9 (0.43) HRH3KDM4EHTTTLR9TLR8
SCHEMBL18980366 0.88 TLR9 (0.43) HRH3KDM4EHTTTLR9TLR8
SCHEMBL18979959 0.87 HRH3 (0.40) HRH3KDM4EHTTKMT2ARAD52
SCHEMBL18980746 0.87 TLR9 (0.42) HRH3TLR9TLR8TLR7L3MBTL3
SCHEMBL21594159 0.83 KDM4E (0.37) HRH3KDM4EHTTKMT2ATLR9
SCHEMBL21594155 0.83 KDM4E (0.37) HRH3KDM4EHTTKMT2ATLR9
SCHEMBL21661577 0.81 KDM4E (0.37) HRH3KDM4EHTTTLR9TLR8
SCHEMBL21661576 0.81 KDM4E (0.37) HRH3KDM4EHTTTLR9TLR8
SCHEMBL18980185 0.81 TLR9 (0.42) IRAK4TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3889146-A1 POLYHETEROCYCLIC TLR7/8 ANTAGONISTS AND THEIR USES FOR TREATING IMMUNE DISORDERS Merck Patent GmbH (DE) 2021-10-06 EP disclosed