SCHEMBL21675259

SCHEMBL21675259

CC(=O)N1c2ccccc2N(C(=O)c2ccc3c(c2)OCO3)CC1C

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.58
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
ALDH1A1 P00352 7/20 0.55
TSHR P16473 6/20 0.55
USP2 O75604 1/20 0.55
LMNA P02545 1/20 0.55
HPGD P15428 3/20 0.54
L3MBTL1 Q9Y468 1/20 0.48
MEN1 O00255 1/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 2/20 0.46
GFER P55789 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16721789 1.00 BRD4 (0.58) BRD4NPC1RAB9AALDH1A1TSHR
SCHEMBL16721360 0.84 BRD4 (0.54) BRD4NPC1RAB9AALDH1A1TSHR
SCHEMBL21675311 0.84 BRD4 (0.54) BRD4NPC1RAB9AALDH1A1TSHR
SCHEMBL21674581 0.82 BRD4 (0.58) BRD4NPC1RAB9ATSHRHPGD
SCHEMBL16721860 0.82 BRD4 (0.58) BRD4NPC1RAB9ATSHRHPGD
SCHEMBL16721973 0.81 BRD4 (0.66) BRD4ALDH1A1HPGDMEN1KMT2A
SCHEMBL16721423 0.81 BRD4 (0.52) BRD4NPC1RAB9AALDH1A1TSHR
SCHEMBL21675133 0.79 BRD4 (0.60) BRD4MEN1KMT2ACYP3A4CYP2C9
SCHEMBL16721785 0.79 BRD4 (0.60) BRD4MEN1KMT2ACYP3A4CYP2C9
SCHEMBL21675261 0.79 BRD4 (0.60) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3071205-B1 BENZOPIPERAZINE COMPOSITIONS AS BET BROMODOMAIN INHIBITORS FORMA THERAPEUTICS INC (US) 2020-02-05 EP disclosed