SCHEMBL21677166

SCHEMBL21677166

CC(C#N)(C#N)CCC(C)(NC(=O)OC(C)(C)C)c1cc(Br)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 13/20 0.45
CTSS P25774 3/20 0.37
CTSK P43235 3/20 0.37
CTSB P07858 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.34
TRPA1 O75762 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18682936 1.00 AAK1 (0.45) AAK1CTSSCTSKCTSBPTGDR2
SCHEMBL18683054 0.85 AAK1 (0.48) AAK1CTSSCTSKPTGDR2NPC1
SCHEMBL18683332 0.84 AAK1 (0.39) AAK1CTSSCTSKCTSBPTGDR2
SCHEMBL21677279 0.84 AAK1 (0.39) AAK1CTSSCTSKCTSBPTGDR2
SCHEMBL18683330 0.84 AAK1 (0.39) AAK1CTSSCTSKCTSBPTGDR2
SCHEMBL21677301 0.84 AAK1 (0.39) AAK1CTSSCTSKCTSBPTGDR2
SCHEMBL27945123 0.83 AAK1 (0.50) AAK1CTSSCTSKPTGDR2NPC1
SCHEMBL253236 0.83 AAK1 (0.50) AAK1CTSSCTSKPTGDR2NPC1
SCHEMBL21677276 0.81 AAK1 (0.42) AAK1CTSSCTSKCTSBTRPA1
SCHEMBL18683317 0.81 AAK1 (0.42) AAK1CTSSCTSKCTSBTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353163-B1 2,3,4,5-TETRAHYDROPYRIDIN-6-AMINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2020-02-05 EP disclosed