SCHEMBL21698765

SCHEMBL21698765

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1ccc(N)nc1)C2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.51
PIK3CA P42336 2/20 0.45
MTOR P42345 2/20 0.45
CYP3A4 P08684 5/20 0.44
ALDH1A1 P00352 4/20 0.44
HIF1A Q16665 3/20 0.44
CYP2C19 P33261 3/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC1 Q13547 1/20 0.44
GPR119 Q8TDV5 4/20 0.43
ACACB O00763 2/20 0.43
USP2 O75604 3/20 0.43
CYP1A2 P05177 3/20 0.43
CYP2C9 P11712 3/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 2/20 0.43
MAPK1 P28482 1/20 0.43
RET P07949 1/20 0.42
TSHR P16473 3/20 0.42
NAMPT P43490 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30664043 0.94 CYP3A4 (0.47) CYP11B2PIK3CAMTORCYP3A4ALDH1A1
SCHEMBL18291310 0.94 CYP3A4 (0.47) CYP11B2PIK3CAMTORCYP3A4ALDH1A1
SCHEMBL20255202 0.93 CYP11B2 (0.48) CYP11B2PIK3CAMTORCYP3A4CYP2C19
SCHEMBL25885002 0.93 CYP11B2 (0.56) CYP11B2PIK3CAMTORALDH1A1HDAC2
SCHEMBL30484800 0.93 CYP11B2 (0.56) CYP11B2PIK3CAMTORALDH1A1HDAC2
SCHEMBL31006174 0.93 CYP11B2 (0.47) CYP11B2PIK3CAMTORCYP3A4ALDH1A1
SCHEMBL19021793 0.93 CYP11B2 (0.47) CYP11B2PIK3CAMTORCYP3A4ALDH1A1
SCHEMBL18291321 0.91 CYP11B2 (0.51) CYP11B2PIK3CAMTORCYP3A4ALDH1A1
SCHEMBL30484809 0.90 CYP11B2 (0.49) CYP11B2PIK3CAMTORALDH1A1HDAC2
SCHEMBL15174881 0.90 CYP11B2 (0.49) CYP11B2PIK3CAMTORALDH1A1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3608321-A1 1H-IMIDAZO[4,5-H]QUINAZOLINE COMPOUND AS PROTEIN KINASE INHIBITOR Shengke Pharmaceuticals (Jiangsu) Ltd. (CN) 2020-02-12 EP disclosed