SCHEMBL2170065

SCHEMBL2170065

CC(C(N)=O)c1ccc(Sc2ccc(F)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
EPHX1 P07099 2/20 0.49
AGBL2 Q5U5Z8 1/20 0.43
APP P05067 1/20 0.42
HTT P42858 2/20 0.41
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
GRM7 Q14831 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
PTPN1 P18031 1/20 0.38
CDC25A P30304 1/20 0.38
CDC25B P30305 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15434305 0.89 EPHX1 (0.58) EPHX1APPHTTALDH1A1GRM7
SCHEMBL2055564 0.89 EPHX1 (0.58) EPHX1APPHTTALDH1A1GRM7
SCHEMBL2170990 0.79 EPHX1 (0.49) EPHX1ALDH1A1
SCHEMBL5677024 0.78 EPHX1 (0.55) EPHX1APPALDH1A1
SCHEMBL22159114 0.76 MEN1 (0.46) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL8427950 0.74 GRM7 (0.45) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL8427951 0.74 GRM7 (0.45) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL8427952 0.74 GRM7 (0.45) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL23003791 0.73 GRM7 (0.47) KMT2AHTTALDH1A1GRM7L3MBTL1
SCHEMBL11469527 0.72 APP (0.49) CYP1A2CYP2C9EPHX1APPMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed