SCHEMBL21702087

SCHEMBL21702087

COc1ccc2[nH]c(C(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](C[C@@H]3CCCNC3=O)C(=O)C(=O)NCc3ccccc3)cc2c1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.53
KDM4E B2RXH2 1/20 0.51
CAPN1 P07384 2/20 0.47
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21702323 0.96 PYGL (0.54) PYGLKDM4ECAPN1CTSLCTSB
SCHEMBL23506377 0.96 PYGL (0.54) PYGLKDM4ECAPN1CTSLCTSB
SCHEMBL21702075 0.92 PYGL (0.53) PYGLCTSLCTSBCTSS
SCHEMBL26493770 0.92 PYGL (0.53) PYGLCTSLCTSBCTSS
SCHEMBL21702080 0.91 PYGL (0.52) PYGLCTSLCTSBCTSS
SCHEMBL23711697 0.91 PYGL (0.52) PYGLCTSLCTSBCTSS
SCHEMBL21702270 0.90 CYP51A1 (0.49)
SCHEMBL26496060 0.90 CYP51A1 (0.49)
SCHEMBL23506504 0.90 CYP51A1 (0.52) PYGL
SCHEMBL21702171 0.90 CYP51A1 (0.52) PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021151387-A1 PHARMACEUTICAL USE OF KETOAMIDE-BASED COMPOUND 中国科学院上海药物研究所 2021-08-05 WO disclosed
EP-3835296-A1 KETOAMIDE COMPOUND AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2021-06-16 EP disclosed
WO-2020030143-A1 KETOAMIDE COMPOUND AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 中国科学院上海药物研究所 2020-02-13 WO disclosed