SCHEMBL2170243

SCHEMBL2170243

CC(C)(CC(=O)NC(COCc1ccccc1)C(=O)Nc1ccc(Oc2ccccc2)cc1)C(N)=O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 13/20 0.62
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TAOK1 Q7L7X3 1/20 0.46
TAOK3 Q9H2K8 1/20 0.46
LTA4H P09960 1/20 0.44
CTSS P25774 1/20 0.43
NPY5R Q15761 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1373995 0.87 S1PR1 (0.68) S1PR1TAOK1TAOK3LTA4H
SCHEMBL2365173 0.85 S1PR1 (0.74) S1PR1SMN1; SMN2NPC1RAB9ATAOK1
SCHEMBL13392751 0.85 S1PR1 (0.73) S1PR1SMN1; SMN2NPC1RAB9ATAOK1
SCHEMBL12044808 0.85 S1PR1 (0.73) S1PR1SMN1; SMN2RAB9ATAOK1TAOK3
SCHEMBL1374371 0.83 S1PR1 (0.68) S1PR1TAOK1TAOK3LTA4H
SCHEMBL1373528 0.83 S1PR1 (0.68) S1PR1SMN1; SMN2NPC1RAB9ATAOK1
SCHEMBL1376155 0.82 S1PR1 (0.73) S1PR1SMN1; SMN2NPC1RAB9ATAOK1
SCHEMBL1373265 0.82 S1PR1 (0.67) S1PR1SMN1; SMN2NPC1RAB9ATAOK1
SCHEMBL12044883 0.82 S1PR1 (0.67) S1PR1SMN1; SMN2NPC1RAB9ATAOK1
SCHEMBL1372544 0.82 S1PR1 (0.67) S1PR1SMN1; SMN2NPC1RAB9ATAOK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed
WO-2010045580-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS EXELIXIS, INC. (US) 2010-04-22 WO disclosed