SCHEMBL21703339

SCHEMBL21703339

Nc1cccn(Cc2nc3ccc(F)cc3n2Cc2ccccc2)c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.50
CYP11B2 P19099 1/20 0.47
AGTR1 P30556 1/20 0.46
AGTR2 P50052 1/20 0.46
RAB9A P51151 1/20 0.46
CD74 P04233 1/20 0.43
MIF P14174 1/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 1/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21684642 0.91 TBXA2R (0.48) AGTR1AGTR2RAB9APLK1TBXA2R
SCHEMBL21703186 0.87 TBXA2R (0.50) AGTR1AGTR2RAB9AKCNK13TBXA2R
SCHEMBL21703232 0.78 MAP4K1 (0.49) BRD4CD74MIFMEN1KMT2A
SCHEMBL21703260 0.78 MAP4K1 (0.49) AGTR1AGTR2RAB9AHTTL3MBTL1
SCHEMBL21702962 0.77 MAP4K1 (0.51) AGTR1AGTR2MEN1KMT2AHTT
SCHEMBL21685620 0.77 ALDH1A1 (0.55) AGTR1AGTR2RAB9ALMNAHTT
SCHEMBL21703340 0.76 MAP4K1 (0.47) AGTR1AGTR2RAB9AMEN1KMT2A
SCHEMBL21703262 0.75 MAP4K1 (0.51) AGTR1AGTR2TBXA2R
SCHEMBL21703266 0.75 MAP4K1 (0.52) AGTR1AGTR2MEN1KMT2ASMN1; SMN2
SCHEMBL21684490 0.75 MAP4K1 (0.48) RAB9ALMNATSHRSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020033784-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS SITARI PHARMA, INC. (US) 2020-02-13 WO disclosed