SCHEMBL2170612

SCHEMBL2170612

CC(C(N)=O)c1ccc(Oc2ccccc2)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.51
PTGS1 P23219 1/20 0.48
LMNA P02545 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PNLIP P16233 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
MEN1 O00255 1/20 0.44
CYP2D6 P10635 1/20 0.44
KMT2A Q03164 1/20 0.44
P2RX4 Q99571 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
XIAP P98170 1/20 0.43
APP P05067 1/20 0.42
ALOX5 P09917 1/20 0.42
CTNNB1 P35222 1/20 0.42
PARG Q86W56 1/20 0.42
STK39 Q9UEW8 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171467 0.89 FFAR1 (0.57) FFAR1PNLIPAPPSTK39ACACB
SCHEMBL2736379 0.81 FFAR1 (0.49) FFAR1PNLIPMRGPRX4PARGSTK39
SCHEMBL2173030 0.79 PARP10 (0.55) FFAR1PTGS1LMNAL3MBTL1MEN1
SCHEMBL7032448 0.78 PTGS1 (0.77) FFAR1PTGS1LMNAL3MBTL1MEN1
SCHEMBL7040469 0.78 PTGS1 (0.77) FFAR1PTGS1LMNAL3MBTL1MEN1
SCHEMBL28775716 0.75 APP (0.55) PTGS1LMNAMEN1KMT2AAKR1C3
SCHEMBL5673527 0.75 APP (0.53) PTGS1LMNAAKR1C3AKR1C2APP
SCHEMBL5673531 0.75 APP (0.53) PTGS1LMNAAKR1C3AKR1C2APP
SCHEMBL30002874 0.75 APP (0.53) PTGS1LMNAAKR1C3AKR1C2APP
SCHEMBL27486876 0.75 PARP10 (0.59) LMNAPNLIPMRGPRX4KMT2ACTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed
WO-2010045580-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS EXELIXIS, INC. (US) 2010-04-22 WO disclosed