SCHEMBL2170743

SCHEMBL2170743

CCCNc1nc(Br)cs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 1/20 0.48
RAB9A P51151 6/20 0.43
MAPT P10636 5/20 0.43
NPC1 O15118 5/20 0.43
ALDH1A1 P00352 4/20 0.43
STAT1 P42224 2/20 0.43
LIMK1 P53667 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HTT P42858 3/20 0.34
PDE7A Q13946 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
NPY5R Q15761 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170914 0.84
SCHEMBL12597147 0.78 RAB9A (0.54) TYRRAB9AMAPTNPC1ALDH1A1
SCHEMBL18398870 0.77 TYR (0.48) TYRRAB9AMAPTNPC1ALDH1A1
SCHEMBL12894438 0.74 TYR (0.46) TYRRAB9AMAPTNPC1ALDH1A1
SCHEMBL217026 0.73
SCHEMBL1747328 0.70 RAB9A (0.81) TYRRAB9AMAPTNPC1ALDH1A1
SCHEMBL12890453 0.68 TYR (0.45) TYRRAB9AMAPTNPC1ALDH1A1
Bromide SCHEMBL1746805 0.67 NPC1 (0.76) TYRRAB9AMAPTNPC1ALDH1A1
SCHEMBL4099165 0.67 RAB9A (0.59) TYRRAB9AMAPTNPC1ALDH1A1
SCHEMBL18398871 0.67 NPC1 (0.51) TYRRAB9AMAPTNPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-27 EP disclosed
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed