SCHEMBL21708870

SCHEMBL21708870

C#CCOC(CN(CC#C)CC#C)c1ccc(O)c(O)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 10/20 0.34
MAPT P10636 9/20 0.34
KDM4E B2RXH2 9/20 0.34
RECQL P46063 7/20 0.34
KMT2A Q03164 5/20 0.34
ADRB2 P07550 5/20 0.34
APEX1 P27695 4/20 0.34
BLM P54132 4/20 0.34
MEN1 O00255 4/20 0.34
DRD2 P14416 4/20 0.34
ADRA1D P25100 4/20 0.34
ADRA1A P35348 4/20 0.34
ADRA1B P35368 4/20 0.34
CYP3A4 P08684 4/20 0.34
ADRB1 P08588 4/20 0.34
ADRB3 P13945 4/20 0.34
MAPK1 P28482 4/20 0.34
LMNA P02545 4/20 0.34
HPGD P15428 3/20 0.34
DRD1 P21728 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709058 0.87 CYP3A4 (0.31) CYP3A4TSHRNFKB1
SCHEMBL21708884 0.80
SCHEMBL21708869 0.80 TDP1 (0.49) TDP1MAPTKDM4ERECQLKMT2A
SCHEMBL21709059 0.80 MAOB (0.32) LMNAHPGDTSHR
SCHEMBL21709085 0.78 PPARG (0.38) TDP1TSHRHIF1AALDH1A1
SCHEMBL21709143 0.77
SCHEMBL21708868 0.75 MAPT (0.41) TDP1MAPTKDM4ERECQLKMT2A
SCHEMBL21708863 0.75 ALOX15 (0.31) TSHRALOX12ALOX15
SCHEMBL21709217 0.72
SCHEMBL21709057 0.70 CYP3A4 (0.40) TDP1MAPTKDM4ERECQLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed