SCHEMBL21709072

SCHEMBL21709072

C#CC(=O)Oc1cc(CCN)ccc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.55
MAPK1 P28482 3/20 0.55
TSHR P16473 2/20 0.55
KDM4E B2RXH2 3/20 0.54
ADRA2A P08913 2/20 0.54
MAPT P10636 2/20 0.54
DRD2 P14416 2/20 0.54
DRD1 P21728 2/20 0.54
DRD4 P21917 2/20 0.54
DRD5 P21918 2/20 0.54
SLC6A2 P23975 2/20 0.54
DRD3 P35462 2/20 0.54
RECQL P46063 2/20 0.54
SLC6A3 Q01959 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
APEX1 P27695 2/20 0.54
ALDH1A1 P00352 1/20 0.54
TP53 P04637 1/20 0.54
ADRB2 P07550 1/20 0.54
HTR1A P08908 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709088 0.89 TSHR (0.47) TAAR1MAPK1TSHRKDM4EADRA2A
SCHEMBL21709073 0.86 TAAR1 (0.50) TAAR1MAPK1TSHRKDM4EADRA2A
SCHEMBL21709089 0.79 TAAR1 (0.52) TAAR1MAPK1TSHRKDM4EADRA2A
SCHEMBL29351887 0.76 TAAR1 (0.55) TAAR1MAPK1TSHRKDM4EADRA2A
SCHEMBL21709064 0.75 TAAR1 (0.58) TAAR1MAPK1TSHRKDM4EADRA2A
Dopamine SCHEMBL9051903 0.73 KDM4E (0.84) TAAR1MAPK1TSHRKDM4EADRA2A
Dopamine SCHEMBL30355306 0.73 KDM4E (0.84) TAAR1MAPK1TSHRKDM4EADRA2A
Dopamine SCHEMBL28995038 0.73 KDM4E (0.84) TAAR1MAPK1TSHRKDM4EADRA2A
Hydrochloric Acid SCHEMBL7360734 0.72 TAAR1 (0.77) TAAR1MAPK1TSHRKDM4EADRA2A
Dopamine SCHEMBL18159501 0.72 KDM4E (1.00) TAAR1MAPK1TSHRKDM4EADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed