SCHEMBL2171406

SCHEMBL2171406

NCc1nc(C(=O)NCCc2cccc(Cl)c2)cs1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.57
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
HTT P42858 1/20 0.57
HIF1A Q16665 2/20 0.55
IGF1R P08069 1/20 0.52
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.51
ADORA2A P29274 1/20 0.51
ADORA1 P30542 1/20 0.51
ALDH1A1 P00352 4/20 0.49
HPGD P15428 1/20 0.49
AKT3 Q9Y243 1/20 0.48
THRB P10828 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
CNR1 P21554 1/20 0.47
IDO1 P14902 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2173104 0.99 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL5670028 0.88 IGF1R (0.56) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL11910629 0.87 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL29698337 0.83 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL24499031 0.83 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL2174354 0.82 HDAC3 (0.52) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL12477893 0.82 IGF1R (0.49) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL5668870 0.81 IGF1R (0.51) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL4390540 0.80 IGF1R (0.52) SMN1; SMN2NPC1RAB9AHTTHIF1A
SCHEMBL2172966 0.80 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9AHTTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730128-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2006-12-13 EP claimed
WO-2005097765-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2005-10-20 WO claimed
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US disclosed
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US disclosed
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US disclosed
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2009-07-23 US disclosed
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2009-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE ALK, BCL3, MCL1 SMN1; SMN2 4564/4885NPC1 1296/4885RAB9A 2862/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.