SCHEMBL21722227

SCHEMBL21722227

Cc1ccc2c(cnn2C2CCCCO2)c1OC(=O)C1CCCCC1=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
CYP4F2 P78329 3/20 0.37
CYP4A11 Q02928 3/20 0.37
POLB P06746 2/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
PDE1A P54750 5/20 0.32
PDE1B Q01064 5/20 0.32
PDE1C Q14123 5/20 0.32
MCL1 Q07820 1/20 0.31
ATR Q13535 1/20 0.30
FGFR1 P11362 1/20 0.30
DDR2 Q16832 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21722547 0.85 RXRA (0.39) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL31510097 0.79 CYP4F2 (0.42) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL27185368 0.79 CYP4F2 (0.42) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL25290373 0.77 RXRA (0.37) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL21722190 0.77 RXRA (0.41) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL27227895 0.75 RXRA (0.47) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL21195792 0.75 CYP4F2 (0.52) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL21230708 0.74 CYP4F2 (0.46) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL18128583 0.74 CYP4F2 (0.44) RXRARXRBRXRGCYP4F2CYP4A11
SCHEMBL21243910 0.74 RXRA (0.38) RXRARXRBRXRGCYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112119075-A Fused ring compound 豪夫迈·罗氏有限公司 2020-12-22 CN disclosed
EP-3746436-A1 FUSED RING COMPOUNDS F. Hoffmann-La Roche AG (CH) 2020-12-09 EP disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed