SCHEMBL21723719

SCHEMBL21723719

COc1c[c]ccc1Nc1nc(C2CC2)c2c(Cl)c[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 7/20 0.42
CLK2 P49760 5/20 0.36
TTK P33981 5/20 0.36
CLK1 P49759 4/20 0.36
CAMKK2 Q96RR4 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
EGFR P00533 1/20 0.35
GAA P10253 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALK Q9UM73 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21723695 0.85 DYRK1A (0.38) LRRK2CLK2TTKCLK1CAMKK2
SCHEMBL28598005 0.84 LRRK2 (0.55) LRRK2CLK2TTKCLK1CAMKK2
SCHEMBL28593022 0.82 LRRK2 (0.54) LRRK2HSP90AA1HSP90AB1KDM4EALDH1A1
SCHEMBL29126151 0.80 HSP90AA1 (0.40) LRRK2HSP90AA1HSP90AB1EGFRKDM4E
SCHEMBL29126098 0.74 LRRK2 (0.40) LRRK2CLK2TTKCLK1CAMKK2
SCHEMBL21738312 0.74 LRRK2 (0.78) LRRK2TTK
SCHEMBL29126132 0.73 EGFR (0.38) LRRK2CLK2TTKCLK1CAMKK2
SCHEMBL21723706 0.72 LRRK2 (0.47) LRRK2EGFR
SCHEMBL21738325 0.71 LRRK2 (0.73) LRRK2TTK
SCHEMBL21738251 0.71 LRRK2 (0.70) LRRK2CLK2TTKCLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020036437-A1 SUBSTITUTED HETEROARYL DERIVATIVE, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING PROTEIN KINASE-RELATED DISEASES WHICH CONTAINS SAME AS ACTIVE INGREDIENT 재단법인 대구경북첨단의료산업진흥재단 2020-02-20 WO claimed
WO-2020036437-A1 SUBSTITUTED HETEROARYL DERIVATIVE, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING PROTEIN KINASE-RELATED DISEASES WHICH CONTAINS SAME AS ACTIVE INGREDIENT 재단법인 대구경북첨단의료산업진흥재단 2020-02-20 WO disclosed