SCHEMBL29126151

SCHEMBL29126151

COc1c[c]ccc1Nc1nc(-c2ccccc2)c2c(Cl)c[nH]c2n1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
LRRK2 Q5S007 7/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EGFR P00533 2/20 0.38
THRB P10828 2/20 0.37
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
ADORA2B P29275 1/20 0.34
ALK Q9UM73 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29126098 0.88 LRRK2 (0.40) HSP90AA1HSP90AB1LRRK2MAPTKDM4E
SCHEMBL28598005 0.84 LRRK2 (0.55) HSP90AA1HSP90AB1LRRK2MAPTKDM4E
SCHEMBL28593022 0.82 LRRK2 (0.54) HSP90AA1HSP90AB1LRRK2MAPTKDM4E
SCHEMBL29126132 0.80 EGFR (0.38) HSP90AA1HSP90AB1LRRK2EGFRJAK2
SCHEMBL28925019 0.80 LRRK2 (0.50) LRRK2MAPTKDM4EALDH1A1KMT2A
SCHEMBL21723719 0.80 LRRK2 (0.42) HSP90AA1HSP90AB1LRRK2MAPTKDM4E
SCHEMBL29126163 0.78 MAPT (0.47) HSP90AA1HSP90AB1LRRK2MAPTKDM4E
SCHEMBL30718282 0.78 MAPT (0.47) HSP90AA1HSP90AB1LRRK2MAPTKDM4E
SCHEMBL30718279 0.73 LRRK2 (0.75) LRRK2
SCHEMBL28925004 0.71 EGFR (0.47) LRRK2EGFRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117247387-A Aromatic heterocyclic compound and preparation method thereof 上海翊石医药科技有限公司 2023-12-19 CN disclosed