SCHEMBL21723720

SCHEMBL21723720

COc1c[c]ccc1Nc1ncc(C(F)(F)F)c(Cl)n1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 15/20 0.48
ALK Q9UM73 2/20 0.43
AURKA O14965 2/20 0.42
KDR P35968 2/20 0.42
AURKB Q96GD4 2/20 0.42
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14995754 0.85 LRRK2 (0.67) LRRK2
SCHEMBL25302280 0.84 LRRK2 (0.50) LRRK2ALK
SCHEMBL2034102 0.83 LRRK2 (0.58) LRRK2ALKAURKAKDRTRPV1
SCHEMBL21723722 0.82 LRRK2 (0.48) LRRK2ALK
SCHEMBL30242558 0.79 LRRK2 (0.56) LRRK2ALKAURKAKDRAURKB
SCHEMBL10206179 0.79 LRRK2 (0.56) LRRK2ALK
SCHEMBL28925066 0.78 LRRK2 (0.58) LRRK2
SCHEMBL14556210 0.78 LRRK2 (0.51) LRRK2ALK
SCHEMBL27897413 0.77 LRRK2 (0.57) LRRK2
SCHEMBL21173791 0.77 TTK (0.57) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020036437-A1 SUBSTITUTED HETEROARYL DERIVATIVE, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING PROTEIN KINASE-RELATED DISEASES WHICH CONTAINS SAME AS ACTIVE INGREDIENT 재단법인 대구경북첨단의료산업진흥재단 2020-02-20 WO disclosed