SCHEMBL21723765

SCHEMBL21723765

O=C(O)N(c1ccc(-c2ccccc2)cc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
OPRK1 P41145 2/20 0.41
UTS2R Q9UKP6 2/20 0.41
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
ESR2 Q92731 1/20 0.41
ACLY P53396 1/20 0.40
PTGER1 P34995 1/20 0.40
PTGER3 P43115 1/20 0.40
PTGER2 P43116 1/20 0.40
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
TSHR P16473 1/20 0.39
CCR2 P41597 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2091976 0.91 NPSR1 (0.47) MEN1KMT2ATSHRNPSR1NPC1
SCHEMBL10569964 0.80 MEN1 (0.43) MEN1KMT2ATSHRHDAC1HDAC6
SCHEMBL2091974 0.79 NPSR1 (0.45) KMT2ATSHRNPSR1NPC1RAB9A
SCHEMBL11438159 0.77 NR3C2 (0.50) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL2092277 0.77 NPC1 (0.43) MEN1KMT2ATSHRNPSR1NPC1
SCHEMBL2095451 0.75 NPSR1 (0.48) MEN1KMT2ATSHRNPSR1NPC1
SCHEMBL8404953 0.74 ALDH1A1 (0.50) KMT2ACYP3A4CYP2D6OPRK1UTS2R
SCHEMBL1942998 0.73 POLQ (0.41) KMT2ATSHRNPSR1NPC1RAB9A
SCHEMBL10344929 0.73 GRM4 (0.43) KMT2ACYP2C9CYP2D6ACLYNPSR1
SCHEMBL29795272 0.73 ALDH1A1 (0.51) MEN1KMT2ANPSR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3836933-A1 INHIBITORS TO TARGET HIV-1 NEF-CD80/CD86 INTERACTIONS FOR THERAPEUTIC INTERVENTION National Centre for Biological Sciences-TIFR (IN) 2021-06-23 EP disclosed
WO-2020035880-A1 INHIBITORS TO TARGET HIV-1 NEF-CD80/CD86 INTERACTIONS FOR THERAPEUTIC INTERVENTION NATIONAL CENTRE FOR BIOLOGICAL SCIENCES-TIFR (IN) 2020-02-20 WO disclosed