SCHEMBL2172659

SCHEMBL2172659

Cc1ccccc1CC(=O)NC(COCc1ccccc1)C(=O)Nc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 14/20 0.66
TAOK1 Q7L7X3 1/20 0.47
TAOK3 Q9H2K8 1/20 0.47
RECQL P46063 1/20 0.45
LTA4H P09960 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1372989 0.91 S1PR1 (0.63) S1PR1TAOK1TAOK3RECQLNPC1
SCHEMBL1375756 0.90 S1PR1 (0.68) S1PR1TAOK1TAOK3RECQLHDAC3
SCHEMBL12044808 0.88 S1PR1 (0.73) S1PR1TAOK1TAOK3RECQLHDAC3
SCHEMBL1373878 0.88 S1PR1 (0.65) S1PR1TAOK1TAOK3RECQLNPC1
SCHEMBL1372558 0.88 S1PR1 (0.67) S1PR1TAOK1TAOK3RECQL
SCHEMBL1373873 0.88 S1PR1 (0.65) S1PR1TAOK1TAOK3RECQLNPC1
SCHEMBL1373394 0.87 S1PR1 (0.67) S1PR1TAOK1TAOK3HDAC3HDAC4
SCHEMBL2365173 0.86 S1PR1 (0.74) S1PR1TAOK1TAOK3RECQLLTA4H
SCHEMBL1374402 0.86 S1PR1 (0.63) S1PR1RECQL
SCHEMBL13392751 0.86 S1PR1 (0.73) S1PR1TAOK1TAOK3RECQLLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed
WO-2010045580-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS EXELIXIS, INC. (US) 2010-04-22 WO disclosed