SCHEMBL21732202

SCHEMBL21732202

Nc1cnc(N2CC(F)(F)CC2c2cccc(F)c2)nc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 3/20 0.44
JAK2 O60674 2/20 0.44
TAAR1 Q96RJ0 1/20 0.39
NOS3 P29474 1/20 0.38
SLC6A9 P48067 3/20 0.36
KDM1A O60341 3/20 0.35
RCOR1 Q9UKL0 1/20 0.35
MAOB P27338 2/20 0.35
MAOA P21397 1/20 0.35
GRM5 P41594 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RIPK1 Q13546 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21723496 0.86 NTRK1 (0.44) NTRK1JAK2NOS3SLC6A9MAOB
SCHEMBL30898796 0.84 NTRK1 (0.47) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL23632045 0.84 NTRK1 (0.47) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL21732293 0.82 NTRK1 (0.46) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL21723165 0.81 NTRK1 (0.47) NTRK1JAK2TAAR1NOS3SLC6A9
SCHEMBL23632049 0.78 NTRK1 (0.45) NTRK1JAK2SLC6A9ALDH1A1MAPT
SCHEMBL21732252 0.78 NTRK1 (0.48) NTRK1JAK2NOS3SLC6A9RIPK1
SCHEMBL21723222 0.78 NTRK1 (0.48) NTRK1JAK2NOS3SLC6A9RIPK1
SCHEMBL21732255 0.78 NTRK1 (0.48) NTRK1JAK2NOS3SLC6A9RIPK1
SCHEMBL448839 0.77 NTRK1 (0.48) NTRK1JAK2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed